Invention Grant
- Patent Title: Compounds as NIK inhibitors
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Application No.: US15520332Application Date: 2015-10-22
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Publication No.: US10005776B2Publication Date: 2018-06-26
- Inventor: George Hynd , Patrizia Tisselli , Janusz Jozef Kulagowski , Calum Macleod , Samuel Edward Mann , Stephen Colin Price , John Gary Montana
- Applicant: Janssen Pharmaceutica NV
- Applicant Address: BE Beerse
- Assignee: Janssen Pharmaceutica NV
- Current Assignee: Janssen Pharmaceutica NV
- Current Assignee Address: BE Beerse
- Priority: EP14190068 20141023
- International Application: PCT/EP2015/074437 WO 20151022
- International Announcement: WO2016/062792 WO 20160428
- Main IPC: A61K31/506
- IPC: A61K31/506 ; C07D471/04

Abstract:
The present invention relates to pharmaceutical agents useful for therapy and/or prophylaxis in a mammal, and in particular to inhibitors of NF-κB-inducing kinase (NIK—also known as MAP3K14) useful for treating diseases such as cancer, inflammatory disorders, metabolic disorders and autoimmune disorders. The invention is also directed to pharmaceutical compositions comprising such compounds, to processes to prepare such compounds and compositions, and to the use of such compounds or pharmaceutical compositions for the prevention or treatment of diseases such as cancer, inflammatory disorders, metabolic disorders including obesity and diabetes, and autoimmune disorders.
Public/Granted literature
- US20170334906A1 NEW COMPOUNDS AS NIK INHIBITORS Public/Granted day:2017-11-23
Information query
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