- Patent Title: Pharmaceutical composition of fused aminodihydrothiazine derivative
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Application No.: US15516567Application Date: 2015-10-08
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Publication No.: US10117876B2Publication Date: 2018-11-06
- Inventor: Yasuhiro Zaima , Kazuo Kazama , Shuntaro Arase , Kentaro Nagane , Kanta Horie , Yosuke Ueki
- Applicant: Eisai R&D Management Co., Ltd.
- Applicant Address: JP Tokyo
- Assignee: Eisai R&D Management Co., Ltd.
- Current Assignee: Eisai R&D Management Co., Ltd.
- Current Assignee Address: JP Tokyo
- Agency: Fish & Richardson P.C.
- Priority: JP2014-209289 20141010
- International Application: PCT/JP2015/078688 WO 20151008
- International Announcement: WO2016/056638 WO 20160414
- Main IPC: A61K31/542
- IPC: A61K31/542 ; C07D513/04 ; A61K9/20

Abstract:
The present invention provides a pharmaceutical composition comprising a compound represented by formula (1): or N-[3-((4aS,5R,7aS)-2-amino-5-methyl-4a,5,7,7a-tetrahydro-4H-furo[3,4-d] [1,3]thiazin-7a-yl)-4-fluorophenyl]-5-difluoromethylpyrazine-2-carboxamide, or a pharmaceutically acceptable salt of the foregoing, and a salt of a compound having a C12-22 saturated aliphatic hydrocarbon group.
Public/Granted literature
- US20180263998A1 PHARMACEUTICAL COMPOSITION OF FUSED AMINODIHYDROTHIAZINE DERIVATIVE Public/Granted day:2018-09-20
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