Invention Grant
- Patent Title: TGR5 agonist complexes for treating diabetes and cancer
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Application No.: US15312157Application Date: 2015-05-26
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Publication No.: US10166246B2Publication Date: 2019-01-01
- Inventor: Donna Yu , James Lester Figarola , Donald David
- Applicant: City of Hope
- Applicant Address: US CA Duarte
- Assignee: City of Hope
- Current Assignee: City of Hope
- Current Assignee Address: US CA Duarte
- Agency: Mintz Levin Cohn Ferris Glovsky and Popeo, P.C.
- International Application: PCT/US2015/032404 WO 20150526
- International Announcement: WO2015/183794 WO 20151203
- Main IPC: A61K31/575
- IPC: A61K31/575 ; A61K31/155 ; C07C279/26 ; C07J9/00 ; C07J41/00 ; C07J63/00 ; A61K31/19

Abstract:
Provided herein are complexes of metformin or metformin analogues and a TGR5 ligand that are useful in treating diseases including diabetes, cardiovascular disease, and cancer.
Public/Granted literature
- US20170196890A1 TGR5 AGONIST COMPLEXES FOR TREATING DIABETES AND CANCER Public/Granted day:2017-07-13
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