• Patent Title: N-acyl-(3-substituted)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor-mediated disorders
  • Application No.: US15956311
    Application Date: 2018-04-18
  • Publication No.: US10214533B2
    Publication Date: 2019-02-26
  • Inventor: Hamid HoveydaGuillaume DutheuilGraeme Fraser
  • Applicant: OGEDA SA
  • Applicant Address: BE Charleroi
  • Assignee: OGEDA SA
  • Current Assignee: OGEDA SA
  • Current Assignee Address: BE Charleroi
  • Agency: Young & Thompson
  • Priority: EP13161864 20130329
  • Main IPC: C07D487/04
  • IPC: C07D487/04 A61K31/4985
N-acyl-(3-substituted)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor-mediated disorders
Abstract:
Novel compounds of Formula I and their use in therapeutic treatments.
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