Invention Grant
- Patent Title: Pyrazolopyrimidine derivatives as NIK inhibitors
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Application No.: US15520346Application Date: 2015-10-22
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Publication No.: US10221180B2Publication Date: 2019-03-05
- Inventor: George Hynd , Patrizia Tisselli , Calum Macleod , Samuel Edward Mann , Terry Aaron Panchal , John Gary Montana , Stephen Colin Price
- Applicant: Janssen Pharmaceutica NV
- Applicant Address: BE Beerse
- Assignee: Janssen Pharmaceutica NV
- Current Assignee: Janssen Pharmaceutica NV
- Current Assignee Address: BE Beerse
- Priority: EP14190073 20141023
- International Application: PCT/EP2015/074431 WO 20151022
- International Announcement: WO2016/062790 WO 20160428
- Main IPC: C07D487/04
- IPC: C07D487/04 ; C07D519/00

Abstract:
The present invention relates to pharmaceutical agents useful for therapy and/or prophylaxis in a mammal, and in particular to inhibitors of NF-κB-inducing kinase (NIK—also known as MAP3K14) useful for treating diseases such as cancer, inflammatory disorders, metabolic disorders and autoimmune disorders. The invention is also directed to pharmaceutical compositions comprising such compounds, to processes to prepare such compounds and compositions, and to the use of such compounds or pharmaceutical compositions for the prevention or treatment of diseases such as cancer, inflammatory disorders, metabolic disorders including obesity and diabetes, and autoimmune disorders.
Public/Granted literature
- US20170334915A1 NEW PYRAZOLOPYRIMIDINE DERIVATIVES AS NIK INHIBITORS Public/Granted day:2017-11-23
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