Invention Grant
- Patent Title: Quinoline derivative
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Application No.: US16540306Application Date: 2019-08-14
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Publication No.: US10676462B2Publication Date: 2020-06-09
- Inventor: Takayuki Inukai , Jun Takeuchi , Tomoko Yasuhiro
- Applicant: ONO PHARMACEUTICAL CO., LTD.
- Applicant Address: JP Osaka
- Assignee: ONO PHARMACEUTICAL CO., LTD.
- Current Assignee: ONO PHARMACEUTICAL CO., LTD.
- Current Assignee Address: JP Osaka
- Agency: Sughrue Mion, PLLC
- Priority: com.zzzhc.datahub.patent.etl.us.BibliographicData$PriorityClaim@2a9a03a7
- Main IPC: C07D401/14
- IPC: C07D401/14 ; C07D215/54 ; C07D401/12

Abstract:
A compound represented by general formula (I) has a strong Axl inhibitory activity by introducing a distinctive bicyclic structure in which a saturated carbon ring is fused to a pyridone ring, and can be a therapeutic agent for Axl-related diseases, for example, cancer such as acute myeloid leukemia, melanoma, breast cancer, pancreatic cancer, and glioma, kidney diseases, immune system diseases, and circulatory system diseases
Public/Granted literature
- US20200002313A1 QUINOLINE DERIVATIVE Public/Granted day:2020-01-02
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