Invention Grant
- Patent Title: Posaconazole, composition, intermediate, preparation method and use thereof
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Application No.: US16081551Application Date: 2016-03-04
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Publication No.: US10696643B2Publication Date: 2020-06-30
- Inventor: Zhiguo Zheng
- Applicant: Zhejiang Ausun Pharmaceutical Co., Ltd.
- Applicant Address: CN Zhejiang
- Assignee: Zhejiang Ausun Pharmaceutical Co., Ltd.
- Current Assignee: Zhejiang Ausun Pharmaceutical Co., Ltd.
- Current Assignee Address: CN Zhejiang
- Agency: Cesari and McKenna, LLP
- International Application: PCT/CN2016/075594 WO 20160304
- International Announcement: WO2017/147893 WO 20170908
- Main IPC: C07D263/26
- IPC: C07D263/26 ; C07D405/14 ; C07D405/06 ; C07D413/06 ; C07D407/06

Abstract:
The present invention relates to a compound of formula III, wherein, R is selected from the group consisting of C1-C4 alkyl, substituted or unsubstituted phenyl, and substituted or unsubstituted benzyl, preferably isopropyl; and two Ar groups may be the same or different, and are each independently selected from the group consisting of substituted or unsubstituted aryl groups, preferably substituted or unsubstituted phenyl, such as p-methoxyphenyl and the like, wherein the compound is preferably in a solid form.
Public/Granted literature
- US20190071408A1 POSACONAZOLE, COMPOSITION, INTERMEDIATE, PREPARATION METHOD THEREFOR, AND USES THEREOF Public/Granted day:2019-03-07
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