Invention Grant
- Patent Title: MU opioid receptor modulators
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Application No.: US15743079Application Date: 2016-06-30
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Publication No.: US10702498B2Publication Date: 2020-07-07
- Inventor: Brian K. Shoichet , Henry Lin , Peter Gmeiner , Aashish Manglik , Brian Kobilka , Bryan L. Roth , Daniela Gisela Dengler
- Applicant: THE REGENTS OF THE UNIVERSITY OF CALIFORNIA , FRIEDRICH-ALEXANDER-UNIVERSITÃT ERLANGEN-NÜRNBERG , THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY , THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL
- Applicant Address: US CA Oakland DE Erlangen US CA Stanford US NC Chapel Hill
- Assignee: THE REGENTS OF THE UNIVERSITY OF CALIFORNIA,FRIEDRICH-ALEXANDER-UNIVERSITAT ERLANGEN-NÜRNBERG,THE BOARD OF TRUSTEES OFTHE LELAND STANFORD JUNIOR UNIVERSITY,THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL
- Current Assignee: THE REGENTS OF THE UNIVERSITY OF CALIFORNIA,FRIEDRICH-ALEXANDER-UNIVERSITAT ERLANGEN-NÜRNBERG,THE BOARD OF TRUSTEES OFTHE LELAND STANFORD JUNIOR UNIVERSITY,THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL
- Current Assignee Address: US CA Oakland DE Erlangen US CA Stanford US NC Chapel Hill
- Agency: Mintz, Levin, Cohn, Ferris, Glovsky and Popeo, P.C.
- Agent Irina E. Britva
- International Application: PCT/US2016/040553 WO 20160630
- International Announcement: WO2017/007695 WO 20170112
- Main IPC: C07C275/26
- IPC: C07C275/26 ; A61K31/381 ; C07D401/12 ; C07C275/24 ; C07D207/452 ; C07D233/16 ; C07D498/18 ; C07D333/16 ; C07D249/04 ; C07D409/12 ; C07D471/04 ; C07D333/20 ; C07D295/125 ; C07D333/58 ; C07D495/04 ; A61P25/36 ; A61K31/165 ; A61K31/17

Abstract:
Described herein, inter alia, are compositions and methods for modulating mu opioid receptor activity.
Public/Granted literature
- US20190076398A1 MU OPIOID RECEPTOR MODULATORS Public/Granted day:2019-03-14
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