Invention Grant
- Patent Title: Processes for the preparation of SGLT-2 inhibitors, intermediates thereof
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Application No.: US15990860Application Date: 2018-05-29
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Publication No.: US10703772B2Publication Date: 2020-07-07
- Inventor: Maha Vishnu Mundla , Sridhar Malyala , Chandra Prakash Narani , Laxmi Narasimha Varaprasad Chintaginjala , Suresh Kumar Gunukula , Bala Yellaiah Chittiboyina , Prabhakar Bellam , Hemalatha Reddy Samireddy , Sowmya Dantham , Prasad Vure , Pooja Kale
- Applicant: Emmennar Pharma Private Limited
- Applicant Address: IN Telangana
- Assignee: Emmennar Pharma Private Limited
- Current Assignee: Emmennar Pharma Private Limited
- Current Assignee Address: IN Telangana
- Agency: Carrier Blackman & Associates, P.C.
- Agent Joseph P. Carrier; Fulchand P. Shende
- Priority: com.zzzhc.datahub.patent.etl.us.BibliographicData$PriorityClaim@264b96cb com.zzzhc.datahub.patent.etl.us.BibliographicData$PriorityClaim@61efc8e8 com.zzzhc.datahub.patent.etl.us.BibliographicData$PriorityClaim@6b1060f8
- Main IPC: A01N43/04
- IPC: A01N43/04 ; A61K31/70 ; C07H7/04 ; C07C41/18 ; C07H7/06 ; A61K47/38 ; C07D307/20 ; A61K9/10 ; A61K9/14

Abstract:
The present invention relates to novel, improved processes for the preparation of sodium glucose co-transporter 2 (SGLT-2) inhibitors and novel intermediates thereof. More particularly, the present invention relates to a novel, improved process for the preparation of gliflozin compounds such as empagliflozin and dapagliflozin, intermediates thereof. The product obtained from the processes of present invention may be amorphous or crystalline, or in the form of amorphous/crystalline solid dispersions/solutions with pharmaceutically acceptable polymers and preparation process thereof. Also, the products obtained from the present invention may be used for the preparation of medicaments for the prevention and/or treatment of diseases and conditions associated with SGLT-2 inhibition.
Public/Granted literature
- US20180346502A1 Processes for the Preparation of SGLT-2 Inhibitors, Intermediates Thereof Public/Granted day:2018-12-06
Information query
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