Invention Grant
- Patent Title: Process for the preparation of dolutegravir
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Application No.: US15549034Application Date: 2016-02-05
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Publication No.: US10730888B2Publication Date: 2020-08-04
- Inventor: Sivaram Prasad Vellanki , Madumurthy Nadella , Mitali Bhalme , Revathi Srinivas Ramabhotla , Venkata Siva Reddy Arumalla , Raveendra Babu Kilaru
- Applicant: Mylan Laboratories Ltd.
- Applicant Address: IN
- Assignee: Mylan Laboratories Limited
- Current Assignee: Mylan Laboratories Limited
- Current Assignee Address: IN
- Priority: com.zzzhc.datahub.patent.etl.us.BibliographicData$PriorityClaim@6345dda5 com.zzzhc.datahub.patent.etl.us.BibliographicData$PriorityClaim@5ebd59fd
- International Application: PCT/IN2016/050046 WO 20160205
- International Announcement: WO2016/125192 WO 20160811
- Main IPC: C07D498/14
- IPC: C07D498/14 ; C07D211/14 ; C07C229/30 ; C07F5/02 ; C07C227/18 ; C07C227/10 ; C07D211/02 ; C07D211/86

Abstract:
Processes for the preparation of dolutegravir and pharmaceutically acceptable salts utilizing alkenylamine are disclosed. Intermediates in those synthetic schemes are also disclosed.
Public/Granted literature
- US20180244693A1 Process for the preparation of dolutegravir Public/Granted day:2018-08-30
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