Invention Grant
- Patent Title: Process for the preparation of phenoxybenzamine
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Application No.: US16478043Application Date: 2018-01-10
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Publication No.: US10906866B2Publication Date: 2021-02-02
- Inventor: Shashi Kant Tiwari , Rajesh Chennuri , Bhanuchandar Samala , Venkata Ramana Kintali , Sivakumaran Meenakshisunderam
- Applicant: AUROBINDO PHARMA LIMITED , Shashi Kant Tiwari , Rajesh Chennuri , Bhanuchandar Samala , Venkata Ramana Kintali , Sivakumaran Meenakshisunderam
- Applicant Address: IN Hyderabad; IN Hyderabad; IN Hyderabad; IN Hyderabad; IN Hyderabad; IN Hyderabad
- Assignee: AUROBINDO PHARMA LIMITED,Shashi Kant Tiwari,Rajesh Chennuri,Bhanuchandar Samala,Venkata Ramana Kintali,Sivakumaran Meenakshisunderam
- Current Assignee: AUROBINDO PHARMA LIMITED,Shashi Kant Tiwari,Rajesh Chennuri,Bhanuchandar Samala,Venkata Ramana Kintali,Sivakumaran Meenakshisunderam
- Current Assignee Address: IN Hyderabad; IN Hyderabad; IN Hyderabad; IN Hyderabad; IN Hyderabad; IN Hyderabad
- Agency: PatentScience LLC
- Agent Jay R. Akhave
- Priority: IN201741001599 20170116
- International Application: PCT/IB2018/050141 WO 20180110
- International Announcement: WO2018/130942 WO 20180719
- Main IPC: C07C213/08
- IPC: C07C213/08

Abstract:
The present invention provides a process for the preparation of N-phenoxyisopropyl ethanolamine of Formula (II) and its conversion to Phenoxybenzamine of Formula (I) or pharmaceutically acceptable salts thereof.
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