Invention Grant
- Patent Title: Inhibitors of protease-activated receptor-2
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Application No.: US16728814Application Date: 2019-12-27
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Publication No.: US10995072B2Publication Date: 2021-05-04
- Inventor: John Graham Cumming , Frank Xinhe Wu , Karl Henrik Edman , Hongming Chen , Dean Gordon Brown , Roland Werner Burli , Shawn Donald Johnstone , Giles Albert Brown , Benjamin Gerald Tehan , Barry John Teobald , Miles Stuart Congreve
- Applicant: Heptares Therapeutics Limited
- Applicant Address: GB Cambridge
- Assignee: Heptares Therapeutics Limited
- Current Assignee: Heptares Therapeutics Limited
- Current Assignee Address: GB Cambridge
- Agency: McCarter & English, LLP
- Agent Steven G. Davis; Mei Bai
- Main IPC: C07D233/64
- IPC: C07D233/64 ; C07D403/06 ; C07D403/10 ; C07D405/06 ; C07D409/06 ; C07D413/10 ; C07D417/10 ; C07D471/04 ; C07D249/08 ; A61P17/00 ; A61P29/00 ; A61K31/4164

Abstract:
The present application relates to certain substituted imidazole compounds, pharmaceutical compositions containing them, and methods of using them, including methods for treating pain, musculoskeletal inflammation, neuroinflammatory disorders, airway inflammation, itch, dermatitis, colitis and related conditions.
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