Invention Grant
- Patent Title: Industrial preparation method for high-purity dicycloplatin needle-like crystal
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Application No.: US16473254Application Date: 2018-06-20
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Publication No.: US10995109B2Publication Date: 2021-05-04
- Inventor: Qinhua Song , Rulin Fan , Jianke Feng
- Applicant: Qinhua Song , Rulin Fan , Jianke Feng
- Applicant Address: CN Jiangsu; CN Jiangsu; CN Jiangsu
- Assignee: Qinhua Song,Rulin Fan,Jianke Feng
- Current Assignee: Qinhua Song,Rulin Fan,Jianke Feng
- Current Assignee Address: CN Jiangsu; CN Jiangsu; CN Jiangsu
- Priority: CN201710472955.0 20170621
- International Application: PCT/CN2018/000229 WO 20180620
- International Announcement: WO2018/233273 WO 20181227
- Main IPC: C07F15/00
- IPC: C07F15/00 ; A61K45/06

Abstract:
Provided is an industrial preparation method for a high-purity dicycloplatin needle-like crystal, comprising: mixing and reacting carboplatin and 1,1-cyclobutane dicarboxylic acid and water, crystallizing same to obtain a dicycloplatin needle-like crystal with a yield of more than 85%, and a utilization rate of the precious metal platinum of more than 97%. The method is green and environmentally friendly and is suitable for industrial production.
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