Invention Grant
- Patent Title: Process for the preparation of 1,5-benzothiazepine compounds
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Application No.: US16545623Application Date: 2019-08-20
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Publication No.: US10995115B2Publication Date: 2021-05-04
- Inventor: Ganapati G. Bhat , Johnson M. Coutinho , Mikael Dahlström , Michael Lofthagen , Akinori Tatara
- Applicant: ELOBIX AB
- Applicant Address: SE Gothenburg
- Assignee: ELOBIX AB
- Current Assignee: ELOBIX AB
- Current Assignee Address: SE Gothenburg
- Agency: Fish & Richardson P.C.
- Priority: IN201811008692 20180309,SE1850474-6 20180423
- Main IPC: C07D281/02
- IPC: C07D281/02 ; C07D281/10 ; C07K5/062

Abstract:
The present invention relates to a process for the preparation of certain 1,5-benzothiazepine compounds, and in particular to a process for the preparation of elobixibat. The process can be carried out under mild and safe conditions and may be used to prepare elobixibat on an industrial scale. The invention also relates to a process for the preparation of a crystalline monohydrate of elobixibat.
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