Invention Grant
- Patent Title: Pharmaceutical composition
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Application No.: US16815183Application Date: 2020-03-11
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Publication No.: US11291661B2Publication Date: 2022-04-05
- Inventor: Geoffrey Gogniat , Saran Kumar , Ulrich Meier , Mario Rentsch
- Applicant: NOVARTIS AG
- Applicant Address: CH Basel
- Assignee: NOVARTIS AG
- Current Assignee: NOVARTIS AG
- Current Assignee Address: CH Basel
- Agent Francine F. Li
- Main IPC: A61K31/46
- IPC: A61K31/46 ; A61P1/16 ; A61K9/00 ; A61K9/16 ; A61K9/20 ; A61K9/28 ; A61K9/48 ; A61K9/50

Abstract:
The present invention relates to the field of pharmacy, particularly to a pharmaceutical composition for oral administration comprising an (a) inert substrate and a (b) mixture comprising a non-bile acid farnesoid X receptor (FXR) agonist, such as 2-[(1R,3r,5S)-3-({5-cyclopropyl-3-[2-(trifluoromethoxy)phenyl]-1,2-oxazol-4-yl}methoxy)-8-azabicyclo[3.2.1]octan-8-yl]-4-fluoro-1,3-benzothiazole-6-carboxylic acid, or a pharmaceutically acceptable salt thereof, and at least one binder. The present invention also relates to a process for preparing said pharmaceutical composition for oral administration; and to the use of said pharmaceutical composition in the manufacture of a medicament.
Public/Granted literature
- US20210169866A1 Pharmaceutical Composition Public/Granted day:2021-06-10
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