Invention Grant
- Patent Title: Prodrugs comprising a pyroglutamate linker
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Application No.: US15577606Application Date: 2016-05-25
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Publication No.: US11298427B2Publication Date: 2022-04-12
- Inventor: Harald Rau , Nicola Bisek , Samuel Weisbrod
- Applicant: Ascendis Pharma A/S , Ascendis Pharma Inc.
- Applicant Address: DK Hellerup; US CA Palo Alto
- Assignee: Ascendis Pharma A/S,Ascendis Pharma Inc.
- Current Assignee: Ascendis Pharma A/S,Ascendis Pharma Inc.
- Current Assignee Address: DK Hellerup; US CA Palo Alto
- Agency: Haug Partners LLP
- Priority: EP15169843 20150529
- International Application: PCT/US2016/034105 WO 20160525
- International Announcement: WO2016/196124 WO 20161208
- Main IPC: A61K47/64
- IPC: A61K47/64 ; A61K47/60 ; A61K47/54

Abstract:
The present invention relates to novel prodrugs of primary or secondary amine-comprising biologically active moieties and pharmaceutically acceptable salts thereof, prodrug reagents, pharmaceutical compositions comprising said prodrugs and the use of prodrugs.
Public/Granted literature
- US20190216940A1 Prodrugs Comprising a Pyroglutamate Linker Public/Granted day:2019-07-18
Information query
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