Invention Grant
- Patent Title: Process for the preparation of linaclotide
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Application No.: US15508928Application Date: 2015-08-29
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Publication No.: US11572386B2Publication Date: 2023-02-07
- Inventor: Suresh Kumar Vadlamani , Patil Nilesh Dagadu , Shafee Mohammed Abdul , Sanjay Devidas Patil , Govindrajan Narayanan
- Applicant: AURO PEPTIDES LTD , Suresh Kumar Vadlamani , Patil Nilesh Dagadu , Shafee Mohammed Abdul , Sanjay Devidas Patil , Govindrajan Narayanan
- Applicant Address: IN Hyderabad; IN Hyderabad; IN Hyderabad; IN Hyderabad; IN Hyderabad; IN Hyderabad
- Assignee: AURO PEPTIDES LTD,Suresh Kumar Vadlamani,Patil Nilesh Dagadu,Shafee Mohammed Abdul,Sanjay Devidas Patil,Govindrajan Narayanan
- Current Assignee: AURO PEPTIDES LTD,Suresh Kumar Vadlamani,Patil Nilesh Dagadu,Shafee Mohammed Abdul,Sanjay Devidas Patil,Govindrajan Narayanan
- Current Assignee Address: IN Hyderabad; IN Hyderabad; IN Hyderabad; IN Hyderabad; IN Hyderabad; IN Hyderabad
- Agency: PatentScience LLC
- Agent Jay R Akhave
- Priority: IN4381/CHE/2014 20140908
- International Application: PCT/IB2015/056555 WO 20150829
- International Announcement: WO2016/038497 WO 20160317
- Main IPC: C07K7/08
- IPC: C07K7/08 ; B01D15/32 ; B01D15/42

Abstract:
The present invention relates to a process for the preparation of Linaclotide by oxidizing linear Linaclotide of formula (II) using combination of air and oxidizing agent followed by purification using RP-HPLC.
Public/Granted literature
- US20170240599A1 A PROCESS FOR THE PREPARATION OF LINACLOTIDE Public/Granted day:2017-08-24
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