Invention Grant
- Patent Title: Process of preparing a peptide epoxyketone immunoproteasome inhibitor, and precursors thereof
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Application No.: US17965064Application Date: 2022-10-13
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Publication No.: US11976053B2Publication Date: 2024-05-07
- Inventor: Henry Johnson , Sean Dalziel , Dustin McMinn
- Applicant: KEZAR LIFE SCIENCES
- Applicant Address: US CA South San Francisco
- Assignee: KEZAR LIFE SCIENCES, INC.
- Current Assignee: KEZAR LIFE SCIENCES, INC.
- Current Assignee Address: US CA South San Francisco
- Agency: MARSHALL, GERSTEIN & BORUN LLP
- The original application number of the division: US17015450 2020.09.09
- Main IPC: C07D295/13
- IPC: C07D295/13 ; C07C229/36 ; C07D295/15 ; C07D301/02 ; C07D303/12 ; C07D303/32 ; C07D303/46

Abstract:
Disclosed herein are methods for preparing [(2S,3R)—N—[(2S)-3-(cyclopent-1-en-1-yl)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]-3-hydroxy-3-(4-methoxyphenyl)-2-[(2S)-2-[2-(morpholin-4-yl)acetamido]propanamido]propanamide (compound “G”):
and precursors thereof.
and precursors thereof.
Public/Granted literature
- US20230135100A1 PROCESS OF PREPARING A PEPTIDE EPOXYKETONE IMMUNOPROTEASOME INHIBITOR, AND PRECURSORS THEREOF Public/Granted day:2023-05-04
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