Invention Grant
- Patent Title: Salts and processes of preparing a PI3K inhibitor
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Application No.: US17365888Application Date: 2021-07-01
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Publication No.: US12024522B2Publication Date: 2024-07-02
- Inventor: Lei Qiao , Lingkai Weng , Chongsheng Eric Shi , David Meloni , Qiyan Lin , Michael Xia , Vaqar Sharief , William Frietze , Zhongjiang Jia , Yongchun Pan , Pingli Liu , Tai-Yuen Yue , Jiacheng Zhou , Jianji Wang
- Applicant: Incyte Corporation
- Applicant Address: US DE Wilmington
- Assignee: Incyte Corporation,Incyte Holdings Corporation
- Current Assignee: Incyte Corporation,Incyte Holdings Corporation
- Current Assignee Address: US DE Wilmington; US DE Wilmington
- Agency: Fish & Richardson P.C.
- The original application number of the division: US15054474 2016.02.26
- Main IPC: C07D487/04
- IPC: C07D487/04

Abstract:
The present application provides processes for preparing (R)-4-(3-((S)-1-(4-amino-3-methyl-1H-pyrazolo[3,4-d]pyrimidin-1-yl)ethyl)-5-chloro-2-ethoxy-6-fluorophenyl)pyrrolidin-2-one, which is useful as an inhibitor phosphoinositide 3-kinase-delta (PI3Kδ), as well as a salt form and intermediates related thereto.
Public/Granted literature
- US20220024934A1 SALTS AND PROCESSES OF PREPARING A PI3K INHIBITOR Public/Granted day:2022-01-27
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