Invention Grant
- Patent Title: Aqueous formulation comprising 1-(4-{[4-(dimethylamino)piperidin-1-yljcarbonyl}phenyl)-3-[4-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)phenyl]urea
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Application No.: US15734147Application Date: 2019-06-04
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Publication No.: US12109308B2Publication Date: 2024-10-08
- Inventor: James Joseph Hussey , Andrew Gilbert Bright
- Applicant: Pfizer Inc.
- Applicant Address: US NY New York
- Assignee: PFIZER INC.
- Current Assignee: PFIZER INC.
- Current Assignee Address: US NY New York
- Agency: Nelson Mullins Riley & Scarborough LLP
- Agent Jane E. Remillard, Esq.; Jill Gorny Sloper, Esq.
- International Application: PCT/IB2019/054643 2019.06.04
- International Announcement: WO2019/234632A 2019.12.12
- Date entered country: 2020-12-01
- Main IPC: A61K9/08
- IPC: A61K9/08 ; A61K9/00 ; A61K9/19 ; A61K31/5377 ; A61K47/02 ; A61K47/12 ; A61K47/26 ; A61K47/40 ; A61P35/00
![Aqueous formulation comprising 1-(4-{[4-(dimethylamino)piperidin-1-yljcarbonyl}phenyl)-3-[4-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)phenyl]urea](/abs-image/US/2024/10/08/US12109308B2/abs.jpg.150x150.jpg)
Abstract:
The present invention relates to a pharmaceutical aqueous formulation comprising 1-(4-{[4-(dimethylamino)piperidin-1-yl]carbonyl}phenyl)-3-[4-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)phenyl]urea, or a pharmaceutically acceptable organic or inorganic acid salt thereof, a pharmaceutically acceptable organic or inorganic acid, a pharmaceutically acceptable beta- or gamma-cyclodextrin and water, that is a clear solution, with the proviso that the organic or inorganic acid (including a salt thereof) is not a sulphonic acid. Such a formulation is particularly suitable for intravenous or parenteral administration to a patient.
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