Invention Grant
US07655690B2 1-sulfonylindole derivatives, their preparation and their use as 5-HT6 ligands
失效
1-磺酰基吲哚衍生物,它们的制备及其作为5-HT6配体的用途
- Patent Title: 1-sulfonylindole derivatives, their preparation and their use as 5-HT6 ligands
- Patent Title (中): 1-磺酰基吲哚衍生物,它们的制备及其作为5-HT6配体的用途
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Application No.: US10566400Application Date: 2004-07-29
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Publication No.: US07655690B2Publication Date: 2010-02-02
- Inventor: Ramon Merce Vidal , Xavier Codony Soler , Alberto Dordal Zueras
- Applicant: Ramon Merce Vidal , Xavier Codony Soler , Alberto Dordal Zueras
- Applicant Address: ES Barcelona
- Assignee: Laboratorios del Dr. Esteve S.A.
- Current Assignee: Laboratorios del Dr. Esteve S.A.
- Current Assignee Address: ES Barcelona
- Agency: Oblon, Spivak, McClelland, Maier & Neustadt, L.L.P.
- Priority: ES200301806 20040730
- International Application: PCT/EP2004/008516 WO 20040729
- International Announcement: WO2005/013974 WO 20050217
- Main IPC: A61K31/415
- IPC: A61K31/415 ; C07D209/04

Abstract:
The present invention refers to new sulfonamide derivatives, of general formula (Ia, Ib, Ic), (I), (Ia, Ib, Ic), optionally in form of one of their stereoisomers, preferably enantiomers or diastereomers, their racemate, or in form of a mixture of at least two of their stereoisomers, preferably enantiomers or diastereomers, in any mixing ratio, or their salts, preferably their corresponding physiologically acceptable salts or corresponding solvates; to the processes for their preparation, to their application as medicaments in human and/or veterinary therapeutics, and to the pharmaceutical compositions containing them. The new compounds of the present invention can be used in the pharmaceutical industry as intermediates and for preparing medicaments.
Public/Granted literature
- US20070060581A1 1-Sulfonylindole derivatives, their preparation and their use as 5-ht6 ligands Public/Granted day:2007-03-15
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