Invention Grant
- Patent Title: Galactose derivative, drug carrier and medicinal composition
- Patent Title (中): 半乳糖衍生物,药物载体和药用组合物
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Application No.: US11574302Application Date: 2005-08-25
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Publication No.: US07655768B2Publication Date: 2010-02-02
- Inventor: Tadaaki Ohgi , Toshihiro Ueda
- Applicant: Tadaaki Ohgi , Toshihiro Ueda
- Applicant Address: JP
- Assignee: Nippon Shinyaku Co., Ltd.
- Current Assignee: Nippon Shinyaku Co., Ltd.
- Current Assignee Address: JP
- Agency: Darby & Darby, P.C.
- Priority: JP2004-246190 20040826
- International Application: PCT/JP2005/015424 WO 20050825
- International Announcement: WO2006/022325 WO 20060302
- Main IPC: C07G3/00
- IPC: C07G3/00 ; C07G11/00 ; C07H15/00 ; C07H17/00 ; A61K31/70 ; A61K9/127 ; A01N43/04

Abstract:
The present invention relates to a novel and useful galactose derivative constituting a drug carrier by which a medicine can be efficiently transferred into the liver, a drug carrier comprising the derivative, and a pharmaceutical composition comprising the carrier and a medicine. The present invention also relates to a galactose derivative made up of galactose, a suitable spacer and a certain lipid, a drug carrier comprising the derivative and a cationic lipid, and a pharmaceutical composition comprising the carrier and a medicine (preferably a double-stranded RNA, a double-stranded DNA, or an oligo nucleic acid).
Public/Granted literature
- US20070244058A1 Galactose Derivative, Drug Carrier and Medicinal Composition Public/Granted day:2007-10-18
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