Invention Grant
- Patent Title: Phthalazinone derivatives
- Patent Title (中): 酞嗪衍生物
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Application No.: US11318155Application Date: 2005-12-23
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Publication No.: US07662818B2Publication Date: 2010-02-16
- Inventor: Niall Morrison Barr Martin , Graeme Cameron Smith , Stephen Philip Jackson , Vincent Junior M Loh , Xiao-Ling Fan Cockcroft , Ian Timothy Williams Matthews , Keith Allan Menear , Frank Kerrigan , Alan Ashworth
- Applicant: Niall Morrison Barr Martin , Graeme Cameron Smith , Stephen Philip Jackson , Vincent Junior M Loh , Xiao-Ling Fan Cockcroft , Ian Timothy Williams Matthews , Keith Allan Menear , Frank Kerrigan , Alan Ashworth
- Applicant Address: GB Cambridge GB Cornwall
- Assignee: Kudos Pharmaceuticals Limited,Maybridge Limited
- Current Assignee: Kudos Pharmaceuticals Limited,Maybridge Limited
- Current Assignee Address: GB Cambridge GB Cornwall
- Agency: Finnegan, Henderson, Farabow, Garrett & Dunner, LLP
- Main IPC: A01N43/60
- IPC: A01N43/60 ; C07D221/02 ; C07D237/30

Abstract:
Compounds of the formula (I): wherein A and B together represent an optionally substituted, fused aromatic ring; X can be NRX or CRXRY; if X=NRX then n is 1 or 2 and if X=CRXRY then n is 1; RX is selected from the group consisting of H, optionally substituted C1-20 alkyl, C5-20 aryl, C3-20 heterocyclyl, amido, thioamido, ester, acyl, and sulfonyl groups; RY is selected from H, hydroxy, amino; or RX and RY may together form a spiro-C3-7 cycloalkyl or heterocyclyl group; RC1 and RC2 are both hydrogen, or when X is CRXRY, RC1, RC2, RX and RY, together with the carbon atoms to which they are attached, may form an optionally substituted fused aromatic ring; and R1 is selected from H and halo.
Public/Granted literature
- US20060149059A1 Phthalazinone derivatives Public/Granted day:2006-07-06
Information query
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