Invention Grant
US07678773B2 Salts of avermectins substituted in the 4″-position and having pesticidal properties 有权
在4“位置取代的除虫菌素的盐具有杀虫性

  • Patent Title: Salts of avermectins substituted in the 4″-position and having pesticidal properties
  • Patent Title (中): 在4“位置取代的除虫菌素的盐具有杀虫性
  • Application No.: US11319687
    Application Date: 2005-12-28
  • Publication No.: US07678773B2
    Publication Date: 2010-03-16
  • Inventor: Thomas Pitterna
  • Applicant: Thomas Pitterna
  • Applicant Address: US GA Duluth
  • Assignee: Merial Limited
  • Current Assignee: Merial Limited
  • Current Assignee Address: US GA Duluth
  • Agency: Merial Limited
  • Agent Judy Jarecki-Black; Thomas Kowalski, Esq.
  • Priority: CH373/01 20010227
  • Main IPC: A61K31/70
  • IPC: A61K31/70 C07H17/08
Salts of avermectins substituted in the 4″-position and having pesticidal properties
Abstract:
A compound of formula wherein X− is an anion; n is 1, 2, 3 or 4; R1 is C1-C12alkyl, C3-C8cycloalkyl; or C2-C12alkenyl; R2 is hydrogen, unsubstituted or substituted C1-C12alkyl or C2-C12alkenyl; R3 is hydrogen, unsubstituted or substituted C1-C12alkyl, C3-C12cycloalkyl, C2-C12alkenyl; or C2-C12alkynyl; or R2 and R3 together are an alkylene or alkenylene bridge; and, where applicable, E/Z isomers, E/Z isomeric mixtures and/or tautomers; with the proviso that R1 is not sec-butyl or isopropyl when R2 is H and R3 is methyl; and, where applicable, their possible tautomers; a process for the preparation of those compounds and their tautomers and the use thereof; pesticidal compositions in which the active ingredient has been selected from those compounds and their tautomers; and a process for the preparation of those compositions and the use thereof; intermediates, in free form or in salt form, for the preparation of those compounds and, where applicable, their tautomers, in free form or in salt form, are described.
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