Invention Grant
US07678912B2 Process for preparation of 4-amino-1-isobutyl-1H-imidazo[4,5-C]-quinoline (Imiquimod) 失效
制备4-氨基-1-异丁基-1H-咪唑并[4,5-C] - 喹啉(咪喹莫特)的方法

Process for preparation of 4-amino-1-isobutyl-1H-imidazo[4,5-C]-quinoline (Imiquimod)
Abstract:
A process for preparation of 1-isobutyl-1H-imidazo-[4,5-c]-quinoline-5-N-oxide, comprising oxidation of 1-isobutyl-1H-imidazoquinoline with meta-chloroperbenzoic acid.
Information query
Patent Agency Ranking
0/0