Invention Grant
- Patent Title: Acetylene derivatives
- Patent Title (中): 乙炔衍生物
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Application No.: US11912626Application Date: 2006-04-24
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Publication No.: US07696379B2Publication Date: 2010-04-13
- Inventor: Ralf Glatthar , Thomas J. Troxler , Thomas Zoller , Joachim Nozulak
- Applicant: Ralf Glatthar , Thomas J. Troxler , Thomas Zoller , Joachim Nozulak
- Applicant Address: CH Basel
- Assignee: Novartis AG
- Current Assignee: Novartis AG
- Current Assignee Address: CH Basel
- Agency: Fanelli, Strain & Haag, PLLC
- Agent Paul D. Strain
- Priority: GB0508319.1 20050425
- International Application: PCT/EP2006/003766 WO 20060424
- International Announcement: WO2006/114262 WO 20061102
- Main IPC: C07C231/00
- IPC: C07C231/00 ; C07D263/02 ; C07D261/02 ; C07D249/08 ; C07D233/00 ; C07C237/00 ; A61K31/33 ; A61K31/16

Abstract:
The invention provides compounds of formula (I) wherein R1 represents hydrogen or alkyl; R2 represents an unsubstituted or substituted heterocycle or R2 represents an unsubstituted or substituted aryl; R3 represents alkyl or halogen; X represents a single bond or an alkandiyl-group, optionally interrupted by one or more oxygen atoms or carbonyl groups or carbonyloxy groups in free base or acid addition salt form, processes for their preparation and their use as pharmaceuticals.
Public/Granted literature
- US20080214673A1 Acetylene Derivatives Public/Granted day:2008-09-04
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