Invention Grant
US07741362B2 Somatostatin receptor 1 and/or 4 selective agonists and antagonists
失效
生长抑素受体1和/或4种选择性激动剂和拮抗剂
- Patent Title: Somatostatin receptor 1 and/or 4 selective agonists and antagonists
- Patent Title (中): 生长抑素受体1和/或4种选择性激动剂和拮抗剂
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Application No.: US10574584Application Date: 2004-10-05
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Publication No.: US07741362B2Publication Date: 2010-06-22
- Inventor: Jussi Tomperi , Paivi Hautamaki , Harri Salo , Mia Engstrom , Andrei Tauber , Anna-Marja Hoffren , Siegfried Wurster
- Applicant: Jussi Tomperi , Paivi Hautamaki , Harri Salo , Mia Engstrom , Andrei Tauber , Anna-Marja Hoffren , Siegfried Wurster
- Applicant Address: FI Piikkio
- Assignee: Siegfried Wurster
- Current Assignee: Siegfried Wurster
- Current Assignee Address: FI Piikkio
- Agency: Oliff & Berridge, PLC
- Priority: FI20031454 20031006
- International Application: PCT/FI2004/000585 WO 20041005
- International Announcement: WO2005/033069 WO 20050414
- Main IPC: A61K31/40
- IPC: A61K31/40 ; A61K31/38 ; A01N41/06 ; A61K31/18 ; C07D209/36 ; C07D333/00
Abstract:
The invention relates to (hetero)arylsulfonylamino based peptidomimetics of formula (I), wherein R1, R2, R3, A, B, D, Q, k and n are defined as disclosed, or a pharmaceutically acceptable salt or ester thereof. Compounds of formula (I) possess high affinity and selectivity for the somatostatin receptor subtypes SSTR1 and/or SSTR4 and can be used for the treatment or diagnosis of diseases or conditions wherein an interaction with SSTR1 and/or SSTR4 is indicated to be useful.
Public/Granted literature
- US20070129422A1 Somatostatin receptor 1 and/or 4 selective agonists and antagonists Public/Granted day:2007-06-07
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