Invention Grant
- Patent Title: Arylindenopyridines and arylindenopyrimidines and related therapeutic and prophylactic methods
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Application No.: US11560637Application Date: 2006-11-16
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Publication No.: US07754730B2Publication Date: 2010-07-13
- Inventor: Geoffrey R. Heintzelman , James Lawrence Bullington , Kenneth C. Rupert
- Applicant: Geoffrey R. Heintzelman , James Lawrence Bullington , Kenneth C. Rupert
- Applicant Address: US NJ Raritan
- Assignee: Ortho-McNeil Pharmaceutical, Inc.
- Current Assignee: Ortho-McNeil Pharmaceutical, Inc.
- Current Assignee Address: US NJ Raritan
- Main IPC: A61K31/505
- IPC: A61K31/505

Abstract:
This invention provides novel arylindenopyridines and arylindenopyrimidines of the formula: wherein R1, R2, R3, R4, and X are as defined above, and pharmaceutical compositions comprising same, useful for treating disorders ameliorated by antagonizing adenosine A2a receptors. This invention also provides therapeutic and prophylactic methods using the instant compounds and pharmaceutical compositions.
Public/Granted literature
- US20070155760A1 ARYLINDENOPYRIDINES AND ARYLINDENOPYRIMIDINES AND RELATED THERAPEUTIC AND PROPHYLACTIC METHODS Public/Granted day:2007-07-05
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