Invention Grant
- Patent Title: Substituted 8-[6-amino-3pyridyl]xanthines
- Patent Title (中): 取代的8- [6-氨基-3-吡啶基]黄嘌呤
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Application No.: US12337010Application Date: 2008-12-17
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Publication No.: US07875608B2Publication Date: 2011-01-25
- Inventor: Robert D. Thompson , Guoquan Wang , Anthony Beauglehole , Frank Schmidtmann
- Applicant: Robert D. Thompson , Guoquan Wang , Anthony Beauglehole , Frank Schmidtmann
- Agency: McCarter & English, LLP
- Main IPC: C07D473/06
- IPC: C07D473/06 ; A61K31/522 ; A61P11/06 ; A61P27/02 ; C07D401/12
![Substituted 8-[6-amino-3pyridyl]xanthines](/abs-image/US/2011/01/25/US07875608B2/abs.jpg.150x150.jpg)
Abstract:
The present invention provides substituted 8-[6-amino-3-pyridyl]xanthines like the compound shown in the following formula: and pharmaceutical compositions that are selective antagonists of A2B adenosine receptors (ARs). These compounds and compositions are useful as pharmaceutical agents.
Public/Granted literature
- US20090163491A1 SUBSTITUTED 8-[6-AMINO-3PYRIDYL]XANTHINES Public/Granted day:2009-06-25
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