Invention Grant
- Patent Title: Heterocyclic janus kinase 3 inhibitors
- Patent Title (中): 杂环janus激酶3抑制剂
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Application No.: US12065234Application Date: 2006-12-25
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Publication No.: US07879844B2Publication Date: 2011-02-01
- Inventor: Takayuki Inoue , Akira Tanaka , Kazuo Nakai , Hiroshi Sasaki , Fumie Takahashi , Shohei Shirakami , Keiko Hatanaka , Yutaka Nakajima , Koichiro Mukoyoshi , Hisao Hamaguchi , Shigeki Kunikawa , Yasuyuki Higashi
- Applicant: Takayuki Inoue , Akira Tanaka , Kazuo Nakai , Hiroshi Sasaki , Fumie Takahashi , Shohei Shirakami , Keiko Hatanaka , Yutaka Nakajima , Koichiro Mukoyoshi , Hisao Hamaguchi , Shigeki Kunikawa , Yasuyuki Higashi
- Applicant Address: JP Tokyo
- Assignee: Astellas Pharma Inc.
- Current Assignee: Astellas Pharma Inc.
- Current Assignee Address: JP Tokyo
- Agency: Oblon, Spivak, McClelland, Maier & Neustadt, L.L.P.
- Priority: JP2005-378858 20051228
- International Application: PCT/JP2006/326327 WO 20061225
- International Announcement: WO2007/077949 WO 20070712
- Main IPC: A61K31/437
- IPC: A61K31/437 ; A61K31/496 ; A61K31/5377 ; A61K31/541 ; C07D471/04 ; C07D471/14 ; A61P37/00 ; A61P25/28 ; A61P35/00

Abstract:
The present invention provides a compound of formula (I) having an excellent JAK3 inhibition activity and being useful as an active ingredient of an agent for treating and/or preventing various immune diseases including autoimmune diseases inflammatory diseases, and allergic diseases. The compound according to the present invention has an inhibition activity against JAK3 and is thus useful as an active ingredient of an agent for treating or preventing diseases caused by undesirable cytokine signal transmission (e.g., rejection during organ/tissue transplantation, autoimmune diseases, multiple sclerosis, rheumatoid arthritis, psoriasis, asthma, atopic dermatitis, Alzheimer's disease, and atherosclerotic disease), or diseases caused by abnormal cytokine signal transmission (e.g., cancer and leukemia).
Public/Granted literature
- US20090270376A1 HETEROCYCLIC JANUS KINASE 3 INHIBITORS Public/Granted day:2009-10-29
Information query
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