Invention Grant
US07919522B2 Compositions comprising C-13 alkoxyether macrolide compounds and phenylpyrazole compounds
有权
包含C-13烷氧基醚大环内酯化合物和苯基吡唑化合物的组合物
- Patent Title: Compositions comprising C-13 alkoxyether macrolide compounds and phenylpyrazole compounds
- Patent Title (中): 包含C-13烷氧基醚大环内酯化合物和苯基吡唑化合物的组合物
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Application No.: US11799796Application Date: 2007-05-03
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Publication No.: US07919522B2Publication Date: 2011-04-05
- Inventor: Mark D. Soll , Albert Boeckh , Natalya Shub
- Applicant: Mark D. Soll , Albert Boeckh , Natalya Shub
- Applicant Address: US GA Duluth
- Assignee: Merial Limited
- Current Assignee: Merial Limited
- Current Assignee Address: US GA Duluth
- Agency: Merial Limited
- Agent Judy Jarecki-Black; John Ezcurra
- Main IPC: A61K31/335
- IPC: A61K31/335 ; C07D309/30
Abstract:
Provided is a novel ivermectin derivative and compositions for the treatment or prophylaxis of parasite infestations in mammals or birds which comprise: (A) a pharmaceutically effective amount of a 1-N-phenylpyrazole compound; (B) a pharmaceutically effective amount of an ivermectin derivative of formula (II) wherein: R14 represents —(CH2)s—O—Z wherein, s is 1 or 2; Y represents —CH(OR15)—, —C(═O)— or —C(═NOR15); R15 represents hydrogen, alkyl or phenyl; and R16 represents —CH3 or —CH2CH3; Z is alkyl, alkenyl, alkynyl, acyl, alkylalkoxy, aryl, alkanoyloxy, alkoxycarbonyl, alkenoyl, alkynoyl, or aroyl.
Public/Granted literature
- US20070293446A1 Compositions comprising C-13 alkoxyether macrolide compounds and phenylpyrazole compounds Public/Granted day:2007-12-20
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