Invention Grant
- Patent Title: Method for the synthesis of peptides without solvent
- Patent Title (中): 无溶剂合成肽的方法
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Application No.: US12531972Application Date: 2008-03-21
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Publication No.: US07960578B2Publication Date: 2011-06-14
- Inventor: Jean Martinez , Frédéric Lamaty , Valérie Declerck
- Applicant: Jean Martinez , Frédéric Lamaty , Valérie Declerck
- Applicant Address: FR Paris FR Montpellier
- Assignee: Centre National de la Recherche Scientifique (CNRS),Universite de Montpellier I
- Current Assignee: Centre National de la Recherche Scientifique (CNRS),Universite de Montpellier I
- Current Assignee Address: FR Paris FR Montpellier
- Agency: Harness, Dickey & Pierce, P.L.C.
- Priority: FR0753970 20070321
- International Application: PCT/EP2008/053444 WO 20080321
- International Announcement: WO2008/125418 WO 20081023
- Main IPC: C07C229/00
- IPC: C07C229/00
Abstract:
The disclosure relates to a method for the synthesis of a compound of the formula (I) in which: n is an integer higher than or equal to 1; Rb and each Rn are independently a hydrogen atom, a C1-C6 arylalkyl group or a C1-C6 alkyl group substituted or not by an aryl group, —COOH, C1-C6, —COO-(alkyl), —CONH2, —SH, heteroaryl, —NH2, —NHC(NH)(NH2), C1-C6-s-(alkyl), —OH or phenol; Ra is a N-protective group; Rc is a ORd group in which Rd is a C1-C6 alkyl group or a NReRf group in which Re and Rf Re independently an N-protective group.
Public/Granted literature
- US20100016631A1 METHOD FOR THE SYNTHESIS OF PEPTIDES WITHOUT SOLVENT Public/Granted day:2010-01-21
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