Invention Grant
- Patent Title: High purity bases of 3,3-diphenylpropylamino monoesters
- Patent Title (中): 3,3-二苯基丙基氨基单酯的高纯度碱
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Application No.: US12141489Application Date: 2008-06-18
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Publication No.: US07989654B2Publication Date: 2011-08-02
- Inventor: Armin Breitenbach , Claus Meese , Hans-Michael Wolff , Roland Drews
- Applicant: Armin Breitenbach , Claus Meese , Hans-Michael Wolff , Roland Drews
- Applicant Address: DE Monheim
- Assignee: UCB Pharma GmbH
- Current Assignee: UCB Pharma GmbH
- Current Assignee Address: DE Monheim
- Agency: Kenyon & Kenyon LLP
- Priority: DE10315917 20030408
- Main IPC: C07C69/017
- IPC: C07C69/017

Abstract:
The invention relates to a compound of general formula (I) wherein A represents deuterium or hydrogen, R represents a group selected from C1-6 alkyl, C3-10 cycloalkyl or phenyl, which can be substituted by C1-3 alkoxy, fluorine, chlorine, bromine, iodine, nitro, amino, hydroxyl, oxo, mercapto or deuterium. The C atom marked with a * (star) can be present in an (R) configuration, in an (S)-configuration or a mixture thereof. The invention is characterized in that the above-mentioned compounds are free bases with a degree of purity of more than 97 wt %. The invention also relates to a method for the production of highly pure compounds of general formula (I) and to the use thereof in the production of medicaments.
Public/Granted literature
- US20090012159A1 HIGH PURITY BASES OF 3,3-DIPHENYLPROPYLAMINO MONOESTERS Public/Granted day:2009-01-08
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