Invention Grant
US08008341B2 Pharmaceutically active benzsulfonamide derivatives as inhibitors of protein junkinases
失效
药物活性苯并磺酰胺衍生物作为蛋白质垃圾酶的抑制剂
- Patent Title: Pharmaceutically active benzsulfonamide derivatives as inhibitors of protein junkinases
- Patent Title (中): 药物活性苯并磺酰胺衍生物作为蛋白质垃圾酶的抑制剂
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Application No.: US12142296Application Date: 2008-06-19
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Publication No.: US08008341B2Publication Date: 2011-08-30
- Inventor: Serge Halazy , Dennis Church , Stephen J. Arkinstall , Marco Biamonte , Montserrat Camps , Jean-Pierre Gotteland , Thomas Rueckle
- Applicant: Serge Halazy , Dennis Church , Stephen J. Arkinstall , Marco Biamonte , Montserrat Camps , Jean-Pierre Gotteland , Thomas Rueckle
- Applicant Address: CH Vaud
- Assignee: Merck Serono SA
- Current Assignee: Merck Serono SA
- Current Assignee Address: CH Vaud
- Agency: Oblon, Spivak, McClelland, Maier & Neustadt, L.L.P.
- Priority: EP00810888 20000927
- Main IPC: A61P25/00
- IPC: A61P25/00 ; A61P37/00 ; A61K31/4468 ; C07D211/96
Abstract:
The present invention relates to benzsulfonamide derivatives of formula I and methods of use thereof. The benzsulfonamide derivatives of the present invention are efficient modulators of the JNK pathway. In particular the benzsulfonamide derivatives of the present invention are selective inhibitors of JNK 2 and 3.
Public/Granted literature
- US20080255222A1 PHARMACEUTICALLY ACTIVE BENZSULFONAMIDE DERIVATIVES AS INHIBITORS OF PROTEIN JUNKINASES Public/Granted day:2008-10-16
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