Invention Grant
- Patent Title: Macrocyclic inhibitors of hepatitis C virus
- Patent Title (中): 丙型肝炎病毒的大环抑制剂
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Application No.: US11995714Application Date: 2006-07-28
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Publication No.: US08012939B2Publication Date: 2011-09-06
- Inventor: Kenneth Alan Simmen , Herman Augustinus De Kock , Pierre Jean-Marie Bernard Raboisson , Sandrine Marie Helene Vendeville , Lili Hu , Abdellah Tahri , Dominique Louis Nestor Ghislain Surleraux , Wim Van De Vreken , Ismet Dorange , Yvan Simonnet , Karl Magnus Nilsson , Bengt Bertil Samuelsson , Asa Annica Kristina Rosenquist , Hans Kristian Wallberg
- Applicant: Kenneth Alan Simmen , Herman Augustinus De Kock , Pierre Jean-Marie Bernard Raboisson , Sandrine Marie Helene Vendeville , Lili Hu , Abdellah Tahri , Dominique Louis Nestor Ghislain Surleraux , Wim Van De Vreken , Ismet Dorange , Yvan Simonnet , Karl Magnus Nilsson , Bengt Bertil Samuelsson , Asa Annica Kristina Rosenquist , Hans Kristian Wallberg
- Applicant Address: IE Cork SE Huddinge
- Assignee: Tibotec Pharmaceuticals Ltd. Co,Medivir AB
- Current Assignee: Tibotec Pharmaceuticals Ltd. Co,Medivir AB
- Current Assignee Address: IE Cork SE Huddinge
- Agent Andrea Jo Kamage
- Priority: EP05107069 20050729
- International Application: PCT/EP2006/064815 WO 20060728
- International Announcement: WO2007/014921 WO 20070208
- Main IPC: A61K38/05
- IPC: A61K38/05 ; C07D245/00

Abstract:
Inhibitors of HCV replication of formula (I) and the N-oxides, salts, and stereoisomers thereof, wherein each variable has specific definitions. Pharmaceutical compositions containing compounds (I) and process for preparing compounds (I) are also provided. Bioavailable combinations of the inhibitors of HCV of Formula (I) with ritonavir are also provided.
Public/Granted literature
- US20090281141A1 MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS Public/Granted day:2009-11-12
Information query
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