Invention Grant
- Patent Title: 2-arylindole derivatives as nPGES-1 inhibitors
- Patent Title (中): 2-芳基吲哚衍生物作为nPGES-1抑制剂
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Application No.: US12306426Application Date: 2007-06-14
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Publication No.: US08017644B2Publication Date: 2011-09-13
- Inventor: Maria Alessandra Alisi , Nicola Cazzolla , Barbara Garofalo , Guido Furlotti , Caterina Maugeri , Rosella Ombrato , Isabella Coletta , Lorenzo Polenzani , Giorgina Mangano , Beatrice Garrone , Angelo Guglielmotti
- Applicant: Maria Alessandra Alisi , Nicola Cazzolla , Barbara Garofalo , Guido Furlotti , Caterina Maugeri , Rosella Ombrato , Isabella Coletta , Lorenzo Polenzani , Giorgina Mangano , Beatrice Garrone , Angelo Guglielmotti
- Applicant Address: IT Rome
- Assignee: Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F. S.p.A.
- Current Assignee: Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F. S.p.A.
- Current Assignee Address: IT Rome
- Agency: Oblon, Spivak, McClelland, Maier & Neustadt, L.L.P.
- Priority: ITMI2006A1368 20060714
- International Application: PCT/EP2007/055901 WO 20070614
- International Announcement: WO2008/006663 WO 20080117
- Main IPC: A61K31/405
- IPC: A61K31/405 ; C07D209/00

Abstract:
A 2-arylindole compound substituted in position 5, of formula (I): in which X, Y, Z, W, A, R and R′ have the meanings given in the description, a pharmaceutical composition comprising it, and also intermediate compounds and a preparation process therefor.
Public/Granted literature
- US20090186922A1 2-ARYLINDOLE DERIVATIVES AS NPGES-I INHIBITORS Public/Granted day:2009-07-23
Information query
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