Invention Grant
US08049038B2 Carnitine conjugates of adamantanamines derivatives as dual prodrugs for various uses 失效
金刚烷胺衍生物的肉碱结合物作为各种用途的双重前药

  • Patent Title: Carnitine conjugates of adamantanamines derivatives as dual prodrugs for various uses
  • Patent Title (中): 金刚烷胺衍生物的肉碱结合物作为各种用途的双重前药
  • Application No.: US13103053
    Application Date: 2011-05-07
  • Publication No.: US08049038B2
    Publication Date: 2011-11-01
  • Inventor: Om P. Goel
  • Applicant: Om P. Goel
  • Applicant Address: US MI Ann Arbor
  • Assignee: SSV Therapeutics, Inc.
  • Current Assignee: SSV Therapeutics, Inc.
  • Current Assignee Address: US MI Ann Arbor
  • Agency: Technology Law, PLLC
  • Agent Karen L. Kimble
  • Main IPC: C07C321/00
  • IPC: C07C321/00
Carnitine conjugates of adamantanamines derivatives as dual prodrugs for various uses
Abstract:
This invention concerns compounds of adamantanamines and neramexane, including their pharmaceutically-acceptable salts, diesterioisomers, and formulations for treating Alzheimer's related dementias, depression, AIDS related dementias, as antivirals, inflammatory diseases such as rheumatoid arthritis, and cerebral ischemia, hyperlipidemia, and diabetes.
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