Invention Grant
US08088779B2 Pyrazolo [1,5-alpha] pyrimidinyl derivatives useful as corticotropin-releasing factor (CRF) receptor antagonists
有权
可用作促肾上腺皮质激素释放因子（CRF）受体拮抗剂的吡唑并[1,5-a]嘧啶基衍生物
![Pyrazolo [1,5-alpha] pyrimidinyl derivatives useful as corticotropin-releasing factor (CRF) receptor antagonists](/docs/US/2012-01-03/US08088779B2/abs.jpg.600x600.jpg)
- Patent Title: Pyrazolo [1,5-alpha] pyrimidinyl derivatives useful as corticotropin-releasing factor (CRF) receptor antagonists
- Patent Title (中): 可用作促肾上腺皮质激素释放因子（CRF）受体拮抗剂的吡唑并[1,5-a]嘧啶基衍生物
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Application No.: US12067939Application Date: 2006-09-28
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Publication No.: US08088779B2Publication Date: 2012-01-03
- Inventor: Frank Hossner
- Applicant: Frank Hossner
- Applicant Address: IE Currabinny, Carrigaline, County Cork
- Assignee: SmithKline Beecham (Cork) Limited
- Current Assignee: SmithKline Beecham (Cork) Limited
- Current Assignee Address: IE Currabinny, Carrigaline, County Cork
- Agent Bonnie L. Deppenbrock
- Priority: GB0519957.5 20050930; WOPCT/US2005/037576 20051019
- International Application: PCT/EP2006/009531 WO 20060928
- International Announcement: WO2007/039264 WO 20070412
- Main IPC: A01N43/90
- IPC: A01N43/90 ; A61K31/519 ; C07D487/00
![Pyrazolo [1,5-alpha] pyrimidinyl derivatives useful as corticotropin-releasing factor (CRF) receptor antagonists](/abs-image/US/2012/01/03/US08088779B2/abs.jpg.150x150.jpg)
Abstract:
The present invention generally relates to the polymorph Form 2 of [3-(4-methoxy-2-methyl-phenyl)-2,5-dimethyl-pyrazolo[1,5-a]pyrimidin-7-yl]-[(S)-1-(3-methyl-[1,2,4]oxa-diazol-5-yl)-propyl]amine. The present invention also relates to pharmaceutical compositions comprising the same and methods of using the same.
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