Invention Grant
US08110579B2 5,6-bisaryl-2-pyridine-carboxamide derivatives, preparation and application thereof in therapeutics as urotensin II receptor antagonists
有权
5,6-二芳基-2-吡啶 - 甲酰胺衍生物,其在治疗剂中的制备及其应用,作为尿素转运蛋白II受体拮抗剂
- Patent Title: 5,6-bisaryl-2-pyridine-carboxamide derivatives, preparation and application thereof in therapeutics as urotensin II receptor antagonists
- Patent Title (中): 5,6-二芳基-2-吡啶 - 甲酰胺衍生物,其在治疗剂中的制备及其应用,作为尿素转运蛋白II受体拮抗剂
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Application No.: US12369200Application Date: 2009-02-11
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Publication No.: US08110579B2Publication Date: 2012-02-07
- Inventor: Jean-Michel Altenburger , Valerie Fossey , Philip Janiak , Gilbert Lassalle , Frederic Petit , Jean Claude Vernieres
- Applicant: Jean-Michel Altenburger , Valerie Fossey , Philip Janiak , Gilbert Lassalle , Frederic Petit , Jean Claude Vernieres
- Applicant Address: FR Paris
- Assignee: Sanofi-Aventis
- Current Assignee: Sanofi-Aventis
- Current Assignee Address: FR Paris
- Agency: Scully, Scott, Murphy & Presser, P.C.
- Priority: FR0607283 20061108
- Main IPC: A61K31/4965
- IPC: A61K31/4965 ; A61K31/444 ; A61K31/4418 ; C07D241/02 ; C07D401/04 ; C07D213/04

Abstract:
The present invention relates to derivatives of 5,6-bisaryl-2-pyridine-carboxamide, their preparation and their application in therapeutics as antagonists of urotensin II receptors.
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