Invention Grant
- Patent Title: Kappa opioid receptor ligands
- Patent Title (中): 卡帕阿片受体配体
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Application No.: US12911244Application Date: 2010-10-25
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Publication No.: US08173678B2Publication Date: 2012-05-08
- Inventor: Frank Ivy Carroll , Hernan A. Navarro , Lawrence E. Brieaddy , Scott P. Runyon , James B. Thomas
- Applicant: Frank Ivy Carroll , Hernan A. Navarro , Lawrence E. Brieaddy , Scott P. Runyon , James B. Thomas
- Applicant Address: US NC Research Triangle Park
- Assignee: Research Triangle Institute
- Current Assignee: Research Triangle Institute
- Current Assignee Address: US NC Research Triangle Park
- Agency: Oblon, Spivak, McClelland, Maier & Neustadt, L.L.P.
- Main IPC: A61K31/451
- IPC: A61K31/451 ; A61K31/453 ; C07D227/06 ; C07D471/18 ; C07D211/18 ; C07D401/12

Abstract:
Kappa opioid receptor antagonists are provided that yield significant improvements in functional binding assays to kappa opioid receptors, and the use of these antagonists in treatment of disease states that are ameliorated by binding of the kappa opioid receptor such as heroin or cocaine addictions.
Public/Granted literature
- US20110065743A1 KAPPA OPIOID RECEPTOR LIGANDS Public/Granted day:2011-03-17
Information query
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