Invention Grant
- Patent Title: Process for preparing Moxifloxacin and salts thereof
- Patent Title (中): 莫西沙星及其盐的制备方法
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Application No.: US13051081Application Date: 2011-03-18
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Publication No.: US08207339B2Publication Date: 2012-06-26
- Inventor: Andrea Castellin , Pierluigi Padovan , Liu Jiageng , Yibo Zhou , Lin Feng
- Applicant: Andrea Castellin , Pierluigi Padovan , Liu Jiageng , Yibo Zhou , Lin Feng
- Applicant Address: IT Alte di Montechhio Maggiore, Vicenza
- Assignee: F.I.S. Fabbrica Italiana Sintetici S.p.A.
- Current Assignee: F.I.S. Fabbrica Italiana Sintetici S.p.A.
- Current Assignee Address: IT Alte di Montechhio Maggiore, Vicenza
- Agency: Dickstein Shapiro LLP
- Priority: ITMI2010A000450 20100319
- Main IPC: C07D471/04
- IPC: C07D471/04
Abstract:
The present invention relates to a process for the synthesis of Moxifloxacin of Formula (I) and salts thereof by means of a process providing the coupling reaction of 1-cyclopropril-6,7-difluoro-1,4-dihydro-8-methoxy-4-oxo -3-quinolinic acid or ester thereof with (4aS, 7aS) -octahydro-1H-pyrrole[3,4-b]pyridine using a magnesium salt.
Public/Granted literature
- US20110230661A1 PROCESS FOR PREPARING MOXIFLOXACIN AND SALTS THEREOF Public/Granted day:2011-09-22
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