Invention Grant
US08212040B2 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and thereof
有权
糖皮质激素模拟物，其制备方法，药物组合物及其制备方法
- Patent Title: Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and thereof
- Patent Title (中): 糖皮质激素模拟物，其制备方法，药物组合物及其制备方法
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Application No.: US11410408Application Date: 2006-04-25
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Publication No.: US08212040B2Publication Date: 2012-07-03
- Inventor: Younes Bekkali , Rajashehar Betageri , Mario G. Cardozo , Thomas A. Gilmore , Christian Hanke Justus Joachim Harcken , Thomas Martin Kirrane , Daniel Kuzmich , John Robert Proudfoot , Doris Riether , Hidenori Takahashi , David S. Thomson , Ji Wang , Renee M. Zindell , Hossein Razavi
- Applicant: Younes Bekkali , Rajashehar Betageri , Mario G. Cardozo , Thomas A. Gilmore , Christian Hanke Justus Joachim Harcken , Thomas Martin Kirrane , Daniel Kuzmich , John Robert Proudfoot , Doris Riether , Hidenori Takahashi , David S. Thomson , Ji Wang , Renee M. Zindell , Hossein Razavi
- Applicant Address: US CT Ridgefield
- Assignee: Boehringer Ingelheim Pharmaceuticals, Inc.
- Current Assignee: Boehringer Ingelheim Pharmaceuticals, Inc.
- Current Assignee Address: US CT Ridgefield
- Agent Michael P. Morris; Timothy X. Witkowski; Usha R. Patel
- Main IPC: C07D471/02
- IPC: C07D471/02 ; A61K31/44
Abstract:
Compounds of Formula (IA) wherein R1, R2, R3, R4 and R5 are as defined herein for Formula (IA), or a tautomer, prodrug, solvate, or salt thereof; pharmaceutical compositions containing such compounds, and methods of modulating the glucocorticoid receptor function and methods of treating disease-states or conditions mediated by the glucocorticoid receptor function or characterized by inflammatory, allergic, or proliferative processes in a patient using these compounds.
Public/Granted literature
- US20060189647A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and thereof Public/Granted day:2006-08-24
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