Invention Grant
US08217172B2 Solid forms of 1-ethyl-3-(5-(5-fluoropyridin-3-yl)-7-(pyrimidin-2-yl)-1H-benzo[d]imidazol-2-yl)urea
失效
固体形式的1-乙基-3-(5-(5-氟吡啶-3-基)-7-(嘧啶-2-基)-1H-苯并[d]咪唑-2-基)脲
- Patent Title: Solid forms of 1-ethyl-3-(5-(5-fluoropyridin-3-yl)-7-(pyrimidin-2-yl)-1H-benzo[d]imidazol-2-yl)urea
- Patent Title (中): 固体形式的1-乙基-3-(5-(5-氟吡啶-3-基)-7-(嘧啶-2-基)-1H-苯并[d]咪唑-2-基)脲
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Application No.: US12329179Application Date: 2008-12-05
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Publication No.: US08217172B2Publication Date: 2012-07-10
- Inventor: Rossitza Alargova , Irina Kadiyala , Arnaud Le Tiran , Dainius Macikenas , Yeugang Zhang
- Applicant: Rossitza Alargova , Irina Kadiyala , Arnaud Le Tiran , Dainius Macikenas , Yeugang Zhang
- Applicant Address: US MA Cambridge
- Assignee: Vertex Pharmaceuticals Incorporated
- Current Assignee: Vertex Pharmaceuticals Incorporated
- Current Assignee Address: US MA Cambridge
- Agent Michael C. Badia
- Main IPC: C07D401/08
- IPC: C07D401/08
![Solid forms of 1-ethyl-3-(5-(5-fluoropyridin-3-yl)-7-(pyrimidin-2-yl)-1H-benzo[d]imidazol-2-yl)urea](/abs-image/US/2012/07/10/US08217172B2/abs.jpg.150x150.jpg)
Abstract:
Solid forms of crystalline1-ethyl-3-(5-(5-fluoropyridin-3-yl)-7-(pyrimidin-2-yl)-1H-benzo[d]imidazol-2-yl)urea, compositions containing solid forms of crystalline1 -ethyl-3-(5-(5-fluoropyridin-3-yl)-7-(pyrimidin-2-yl)-1H-benzo[d]imidazol-2-yl)urea and methods of using the same are described.
Public/Granted literature
- US20100063284A1 SOLID FORMS OF 1-ethyl-3-(5-(5-FLUOROPYRIDIN-3-YL)-7-(PYRIMIDIN-2-YL)-1H-BENZO[D]IMIDAZOL-2-YL)UREA Public/Granted day:2010-03-11
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