Invention Grant
- Patent Title: Process for preparing macrocyclic compounds
- Patent Title (中): 制备大环化合物的方法
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Application No.: US12552569Application Date: 2009-09-02
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Publication No.: US08222369B2Publication Date: 2012-07-17
- Inventor: Carl Alan Busacca , Fabrice Gallou , Nizar Haddad , Azad Hossain , Suresh R. Kapadia , Jianxiu Liu , Chris H. Senanayake , Xudong Wei , Nathan K. Yee
- Applicant: Carl Alan Busacca , Fabrice Gallou , Nizar Haddad , Azad Hossain , Suresh R. Kapadia , Jianxiu Liu , Chris H. Senanayake , Xudong Wei , Nathan K. Yee
- Applicant Address: DE Ingelheim am Rhein
- Assignee: Boehringer Ingelheim International GmbH
- Current Assignee: Boehringer Ingelheim International GmbH
- Current Assignee Address: DE Ingelheim am Rhein
- Agent Michael P. Morris; Philip I. Datlow
- Main IPC: C07K1/00
- IPC: C07K1/00

Abstract:
Disclosed is a process for preparing a macrocyclic compound of the formula (I) wherein a hydroxyl-substituted macrocyclic compound of formula (3) is reacted with a sulfonyl-substituted compound of formula QUIN: The compounds of formula (I) are potent active agents for the treatment of hepatitis C virus (HCV) infection.
Public/Granted literature
- US20090326194A1 PROCESS FOR PREPARING MACROCYCLIC COMPOUNDS Public/Granted day:2009-12-31
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