Invention Grant
- Patent Title: Heterocyclic inhibitors of stearoyl-CoA desaturase
- Patent Title (中): 硬脂酰辅酶A去饱和酶的杂环抑制剂
-
Application No.: US12442279Application Date: 2007-09-19
-
Publication No.: US08236835B2Publication Date: 2012-08-07
- Inventor: Natalie Dales , Zaihui Zhang , Rajender Kamboj , Jianmin Fu , Shaoyi Sun , Natalia Pokrovskaia , Serguei Sviridov
- Applicant: Natalie Dales , Zaihui Zhang , Rajender Kamboj , Jianmin Fu , Shaoyi Sun , Natalia Pokrovskaia , Serguei Sviridov
- Applicant Address: CH Basel CA Burnaby
- Assignee: Novartis AG,Xenon Pharmaceuticals Inc.
- Current Assignee: Novartis AG,Xenon Pharmaceuticals Inc.
- Current Assignee Address: CH Basel CA Burnaby
- Agent Joshua Roth
- International Application: PCT/US2007/078854 WO 20070919
- International Announcement: WO2008/036715 WO 20080327
- Main IPC: A61K31/426
- IPC: A61K31/426

Abstract:
The present invention provides heterocyclic derivatives that modulate the activity of stearoyl-CoA desaturase. Methods of using such derivatives to modulate the activity of stearoyl-CoA desaturase and pharmaceutical compositions comprising such derivatives are also encompassed.
Public/Granted literature
- US20100029718A1 ORGANIC COMPOUNDS Public/Granted day:2010-02-04
Information query
IPC分类: