Invention Grant
US08258129B2 4-heterocycloalkylpyri(mi)dines, process for the preparation thereof and their use as medicaments
有权
4-杂环烷基吡啶(mi)餐,其制备方法及其作为药物的用途
- Patent Title: 4-heterocycloalkylpyri(mi)dines, process for the preparation thereof and their use as medicaments
- Patent Title (中): 4-杂环烷基吡啶(mi)餐,其制备方法及其作为药物的用途
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Application No.: US12304134Application Date: 2007-07-05
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Publication No.: US08258129B2Publication Date: 2012-09-04
- Inventor: Harald Engelhardt , Gerd Bader , Guido Boehmelt , Ralph Brueckner , Thomas Gerstberger , Maria Impagnatiello , Daniel Kuhn , Otmar Schaaf , Heinz Stadtmueller , Irene Waizenegger , Andreas Zoephel
- Applicant: Harald Engelhardt , Gerd Bader , Guido Boehmelt , Ralph Brueckner , Thomas Gerstberger , Maria Impagnatiello , Daniel Kuhn , Otmar Schaaf , Heinz Stadtmueller , Irene Waizenegger , Andreas Zoephel
- Applicant Address: DE Ingelheim am Rhein
- Assignee: Boehringer Ingelheim International GmbH
- Current Assignee: Boehringer Ingelheim International GmbH
- Current Assignee Address: DE Ingelheim am Rhein
- Agent Michael P. Morris; Alan R. Stempel
- Priority: EP06116748 20060706
- International Application: PCT/EP2007/056853 WO 20070705
- International Announcement: WO2008/003766 WO 20080110
- Main IPC: C07D471/04
- IPC: C07D471/04 ; C07D487/04 ; A61K31/506

Abstract:
The present invention encompasses compounds of general formula (1) wherein X and R1 to R3 are as defined in the disclosure, which are suitable for the treatment of diseases characterized by excessive or abnormal cell proliferation, and the use thereof for preparing a pharmaceutical composition having the above-mentioned properties.
Public/Granted literature
- US20090203673A1 4-HETEROCYCLOALKYLPYRI(MI)DINES, PROCESS FOR THE PREPARATION THEREOF AND THEIR USE AS MEDICAMENTS Public/Granted day:2009-08-13
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