Invention Grant
US08258308B2 Amino nicotinic and isonicotinic acid derivatives as DHODH inhibitors
有权
氨基烟碱和异烟酸衍生物作为DHODH抑制剂
- Patent Title: Amino nicotinic and isonicotinic acid derivatives as DHODH inhibitors
- Patent Title (中): 氨基烟碱和异烟酸衍生物作为DHODH抑制剂
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Application No.: US12520237Application Date: 2007-12-21
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Publication No.: US08258308B2Publication Date: 2012-09-04
- Inventor: Julio Cesar Castro Palomino Laria , Montserrat Erra Sola , Maria Estrella Lozoya Toribio , Eloisa Navarro Romero
- Applicant: Julio Cesar Castro Palomino Laria , Montserrat Erra Sola , Maria Estrella Lozoya Toribio , Eloisa Navarro Romero
- Applicant Address: ES Barcelona
- Assignee: Laboratorios Almirall, S.A.
- Current Assignee: Laboratorios Almirall, S.A.
- Current Assignee Address: ES Barcelona
- Agency: Finnegan, Henderson Farabow, Garrett & Dunner, LLP
- Priority: ES200603250 20061222; ES200701086 20070423
- International Application: PCT/EP2007/011401 WO 20071221
- International Announcement: WO2008/077639 WO 20080703
- Main IPC: C07D211/78
- IPC: C07D211/78 ; C07D213/79 ; C07D421/00 ; A61K31/44

Abstract:
The present disclosure relates to compounds of formula (I): or a pharmaceutically acceptable salt or N-oxide thereof. The present disclosure also relates to pharmaceutical compositions comprising the compounds of formula (I), and to their methods of use in therapy.
Public/Granted literature
- US20100074898A1 AMINO NICOTINIC AND ISONICOTINIC ACID DERIVATIVES AS DHODH INHIBITORS Public/Granted day:2010-03-25
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