Invention Grant
US08378097B2 3-(1,3-benzodioxol-5-yl)-6-(4-cyclopropylpiperazin-1-yl)-pyridazine, its salts and solvates and its use as histamine H3 receptor antagonist 有权
3-(1,3-苯并间二氧杂环戊烯-5-基)-6-(4-环丙基哌嗪-1-基) - 哒嗪及其盐和溶剂合物及其作为组胺H3受体拮抗剂

  • Patent Title: 3-(1,3-benzodioxol-5-yl)-6-(4-cyclopropylpiperazin-1-yl)-pyridazine, its salts and solvates and its use as histamine H3 receptor antagonist
  • Patent Title (中): 3-(1,3-苯并间二氧杂环戊烯-5-基)-6-(4-环丙基哌嗪-1-基) - 哒嗪及其盐和溶剂合物及其作为组胺H3受体拮抗剂
  • Application No.: US12302132
    Application Date: 2007-05-22
  • Publication No.: US08378097B2
    Publication Date: 2013-02-19
  • Inventor: Rolf Hohlweg
  • Applicant: Rolf Hohlweg
  • Applicant Address: US NC High Point
  • Assignee: High Point Pharmaceuticals, LLC
  • Current Assignee: High Point Pharmaceuticals, LLC
  • Current Assignee Address: US NC High Point
  • Agent Samuel B. Rollins
  • Priority: EP06114615 20060529; EP06120117 20060905
  • International Application: PCT/EP2007/054940 WO 20070522
  • International Announcement: WO2007/137968 WO 20071206
  • Main IPC: C07D237/02
  • IPC: C07D237/02 A61K31/50
3-(1,3-benzodioxol-5-yl)-6-(4-cyclopropylpiperazin-1-yl)-pyridazine, its salts and solvates and its use as histamine H3 receptor antagonist
Abstract:
3-(1,3-Benzodioxol-5-yl)-6-(4-cyclopropylpiperazin-1-yl)pyridazine and salts and solvates thereof, having histamine H3 antagonistic activity can be used in pharmaceutical compositions.
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