Invention Grant
- Patent Title: Macrolides and their use
- Patent Title (中): 大环内酯类及其用途
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Application No.: US12864921Application Date: 2009-02-09
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Publication No.: US08410065B2Publication Date: 2013-04-02
- Inventor: Johannes Laurenz Kellenberger , Jürg Dreier , Stefan Bernhard Reinelt
- Applicant: Johannes Laurenz Kellenberger , Jürg Dreier , Stefan Bernhard Reinelt
- Applicant Address: CH Basel
- Assignee: Basilea Pharmaceutica AG
- Current Assignee: Basilea Pharmaceutica AG
- Current Assignee Address: CH Basel
- Priority: EP08101438 20080208
- International Application: PCT/EP2009/051441 WO 20090209
- International Announcement: WO2009/106419 WO 20090903
- Main IPC: A61K31/70
- IPC: A61K31/70 ; C07H17/08

Abstract:
The invention relates to antibiotic macrolides of formula (I), which have improved anti-inflammatory activity mediated through inhibition of phosphodiesterase 4 (PDE4) useful for the treatment and/or prevention of inflammatory, allergic and proliferative diseases.
Public/Granted literature
- US20110053876A1 MACROLIDES AND THEIR USE Public/Granted day:2011-03-03
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