Invention Grant
- Patent Title: Pyrrolidin-2-one derivatives as androgen receptor modulator
- Patent Title (中): 吡咯烷-2-酮衍生物作为雄激素受体调节剂
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Application No.: US12672516Application Date: 2008-08-06
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Publication No.: US08420694B2Publication Date: 2013-04-16
- Inventor: Atsushi Hasuoka
- Applicant: Atsushi Hasuoka
- Applicant Address: JP Osaka
- Assignee: Takeda Pharmaceutical Company Limited
- Current Assignee: Takeda Pharmaceutical Company Limited
- Current Assignee Address: JP Osaka
- Agency: Edwards Wildman Palmer LLP
- Agent David G. Conlin; Mark D. Russett
- Priority: JP2007-205966 20070807; JP2007-299658 20071119
- International Application: PCT/JP2008/064500 WO 20080806
- International Announcement: WO2009/020234 WO 20090212
- Main IPC: A61K31/40
- IPC: A61K31/40 ; C07D207/00

Abstract:
A compound represented by the formula (I′): or a salt thereof, has a superior androgen modulating action, wherein R1, R2, R4 to R8, R10 and R11 are defined in the claim.
Public/Granted literature
- US20110098336A1 PYRROLIDIN-2-ONE DERIVATIVES AS ANDROGEN RECEPTOR MODULATOR Public/Granted day:2011-04-28
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